{"product_id":"blood-brain-barrier-in-drug-discovery-li-di-9781118788356","title":"Blood-Brain Barrier in Drug Discovery: Optimizing Brain Exposure of CNS Drugs and Minimizing Brain Side Effects for Peripheral Drugs","description":"\u003cp\u003eFocused on central nervous system (CNS) drug discovery efforts, this book educates drug researchers about the blood-brain barrier (BBB) so they can affect important improvements in one of the most significant - and most challenging - areas of drug discovery.\u003c\/p\u003e \u003cp\u003e- Written by world experts to provide practical solutions to increase brain penetration or minimize CNS side-effects\u003cbr\u003e - Reviews state-of-the-art in silico, in vitro, and in vivo tools to assess brain penetration and advanced CNS drug delivery strategies\u003cbr\u003e - Covers BBB physiology, medicinal chemistry design principles, free drug hypothesis for the BBB, and transport mechanisms including passive diffusion, uptake\/efflux transporters, and receptor-mediated processes\u003cbr\u003e - Highlights the advances in modelling BBB pharmacokinetics and dynamics relationships (PK\/PD) and physiologically-based pharmacokinetics (PBPK)\u003cbr\u003e - Discusses case studies of successful CNS and non-CNS drugs, lessons learned and paths to the market\u003c\/p\u003e\u003cbr\u003e\u003cbr\u003e\u003cb\u003eAuthor:\u003c\/b\u003e Li Di\u003cbr\u003e\u003cb\u003eISBN-10:\u003c\/b\u003e 1118788354\u003cbr\u003e\u003cb\u003eISBN-13:\u003c\/b\u003e 9781118788356\u003cbr\u003e\u003cb\u003ePublisher:\u003c\/b\u003e Wiley\u003cbr\u003e\u003cb\u003eLanguage:\u003c\/b\u003e English\u003cbr\u003e\u003cb\u003ePublished:\u003c\/b\u003e 02\/09\/2015\u003cbr\u003e\u003cb\u003ePages:\u003c\/b\u003e 608\u003cbr\u003e\u003cb\u003eFormat:\u003c\/b\u003e Hardcover\u003cbr\u003e\u003cb\u003eWeight:\u003c\/b\u003e 2.02lbs\u003cbr\u003e\u003cb\u003eSize:\u003c\/b\u003e 9.30h x 6.30w x 1.40d","brand":"Li Di","offers":[{"title":"Hardcover","offer_id":43980865962239,"sku":"9781118788356","price":166.95,"currency_code":"USD","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0662\/2982\/9887\/files\/img_7b775e03-784a-44f5-925c-72f55252310d.jpg?v=1683252339","url":"https:\/\/www.whiterainbookhouse.com\/products\/blood-brain-barrier-in-drug-discovery-li-di-9781118788356","provider":"WR Book House","version":"1.0","type":"link"}